Serine/threonine-protein kinase/endoribonuclease IRE1

Basic Information


Uniprot ID: O75460
Secondary ID: A1L457
Symbol: ERN1
Other Name: IRE1,Endoplasmic reticulum-to-nucleus signaling 1,Inositol-requiring protein 1,hIRE1p,Ire1-alpha,IRE1a
Class: Single Protein
Type: pro-fibrotic
Molecular Function: Hydrolase,Kinase,Multifunctional enzyme,Serine/threonine-protein kinase,Transferase


Target Classification


Category I Category II Category III
Intracellular Enzyme Kinase

Related Compound


Target ID Name Interaction
D0516 3,6-DMAD inhibitor

Fibrosis Related Property


Reference Record 1

PubMed ID 29316036 Compound ID D0516
CAS Name 3,6-DMAD
Model vitro,mice Fibrosis Disease Keloid
Process I
Process II
Process III prevenet collagen deposition
Mechanism