Cytosolic phospholipase A2

Basic Information


Uniprot ID: P47712
Secondary ID: B1AKG4, Q29R80
Symbol: PLA2G4A
Other Name: CPLA2,cPLA2,Phospholipase A2 group IVA,Phosphatidylcholine 2-acylhydrolase
Class: Single Protein
Type: pro-fibrotic
Molecular Function: Hydrolase


Target Classification


Category I Category II Category III
Intracellular Enzyme Hydrolase

Related Compound


Target ID Name Interaction
D0396 Arachidonyl trifluoro-methyl-ketone inhibitor

Fibrosis Related Property


Reference Record 1

PubMed ID 26045535 Compound ID
CAS Name
Model mice Fibrosis Disease Renal fibrosis
Process I attenue inflammation
Process II
Process III prevenet collagen deposition
Mechanism

Reference Record 2

PubMed ID 22093332 Compound ID
CAS Name
Model vitro Fibrosis Disease Liver fibrosis
Process I
Process II HSCs activation
Process III
Mechanism Targeting PPAR-β/δ signaling

Reference Record 3

PubMed ID 20429932 Compound ID D0396
CAS 149301-79-1 Name Arachidonyl trifluoro-methyl-ketone
Model mice Fibrosis Disease Cystic fibrosis
Process I
Process II
Process III
Mechanism

Reference Record 4

PubMed ID 20413542 Compound ID
CAS Name
Model vitro,mice Fibrosis Disease Cystic fibrosis
Process I
Process II
Process III
Mechanism