C5a anaphylatoxin chemotactic receptor 1

Basic Information


Uniprot ID: P21730
Secondary ID:
Symbol: C5AR1
Other Name: C5AR,C5a anaphylatoxin chemotactic receptor,C5a-R,C5aR,
Class: Single Protein
Type: pro-fibrotic
Molecular Function: G-protein coupled receptor,Receptor,Transducer


Target Classification


Category I Category II Category III
Extracellular G protein-coupled receptor Other peptide receptor

Related Compound


Target ID Name Interaction
D0208 W-54011 antagonist
D0450 JPE-1375 antagonist

Fibrosis Related Property


Reference Record 1

PubMed ID 26001927 Compound ID D0208
CAS 405098-33-1 Name W-54011
Model vitro,mice Fibrosis Disease Pancreatic fibrosis
Process I
Process II fibroblasts activation
Process III prevenet collagen deposition
Mechanism

Reference Record 2

PubMed ID 17389734 Compound ID D0450
CAS Name JPE-1375
Model vitro Fibrosis Disease Renal fibrosis
Process I
Process II
Process III prevenet collagen deposition
Mechanism