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Histone deacetylases
Basic Information
Uniprot ID:
Secondary ID:
Symbol:
Other Name:
Class:
Protein Famliy
Type:
pro-fibrotic
Molecular Function:
Target Classification
Category I
Category II
Category III
Other
Related Compound
Target ID
Name
Interaction
D0133
Vorinostat
inhibitor
D0159
Givinostat
inhibitor
D0275
HNHA
inhibitor
Fibrosis Related Property
Reference Record 1
PubMed ID
27367506
Compound ID
D0133
CAS
149647-78-9
Name
Vorinostat
Model
rabbit
Fibrosis Disease
Scar
Process I
Process II
Process III
prevenet collagen deposition
Mechanism
Reference Record 2
PubMed ID
26865052
Compound ID
D0159
CAS
497833-27-9
Name
Givinostat
Model
vitro,rabbit
Fibrosis Disease
Corneal fibrosis
Process I
Process II
fibroblasts differetiation,fibroblast migration
Process III
prevenet collagen deposition
Mechanism
Targeting TGFβ/BMP7 signaling pathway
Reference Record 3
PubMed ID
24467283
Compound ID
D0275
CAS
926908-04-5
Name
HNHA
Model
vitro,mice,rat
Fibrosis Disease
Liver fibrosis
Process I
Process II
HSCs activation,HSCs proliferation,HSCs apoptosis
Process III
prevenet collagen deposition
Mechanism