Nuclear receptor subfamily 1 group D member 1

Basic Information


Uniprot ID: P20393
Secondary ID: Q0P5Z4, Q15304
Symbol: NR1D1
Other Name: EAR1,Rev-erbA-alpha,V-erbA-related protein 1,EAR-1
Class: Single Protein
Type: pro-fibrotic
Molecular Function: Activator,DNA-binding,Receptor,Repressor


Target Classification


Category I Category II Category III
Intracellular Nuclear receptor NR1 family

Related Compound


Target ID Name Interaction
D0269 SR6452 modulator
D0521 SR8278 antagonist

Fibrosis Related Property


Reference Record 1

PubMed ID 24497272 Compound ID D0269
CAS 1216744-19-2 Name SR6452
Model vitro,human,rat Fibrosis Disease Liver fibrosis
Process I
Process II HSCs activation
Process III prevenet collagen deposition
Mechanism

Reference Record 2

PubMed ID 29215066 Compound ID D0521
CAS 1254944-66-5 Name SR8278
Model vitro,mice Fibrosis Disease Muscle fibrosis
Process I
Process II cells activation,cells differentiation
Process III prevenet collagen deposition
Mechanism