Bioactive Compounds List
Type Distribution
Max Phase Distribution
Bioactive Compounds List
| Bio ID | Target ID | Target Name | ChEMBL ID | Name | Type | Max Phase | Molecular Weight | Targets | Bioactivities | Molecular Formula | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|
| bio1991 | Tar12 | Toll-like receptor 9 (TLR9) | CHEMBL3544947 | BURAPITANT | Small molecule | Phase 2 | 682.53 | -- | -- | C31H35Cl2F6N3O3 | Details |
| bio1992 | Tar12 | Toll-like receptor 9 (TLR9) | CHEMBL573677 | ABEQUOLIXRON | Small molecule | Phase 1 | 596.09 | 6.0 | 20.0 | C34H33ClF3NO3 | Details |
| bio1993 | Tar12 | Toll-like receptor 9 (TLR9) | CHEMBL4297922 | TUMOR NECROSIS FACTOR RECEPTOR SUPERFAMILY MEMBER 9 | Unknown | Phase 1 | -- | -- | -- | -- | Details |
| bio1994 | Tar12 | Toll-like receptor 9 (TLR9) | CHEMBL3989695 | REGADENOSON | Small molecule | Phase 4 | 408.38 | -- | -- | C15H20N8O6 | Details |
| bio1995 | Tar12 | Toll-like receptor 9 (TLR9) | CHEMBL1201284 | CINACALCET | Small molecule | Phase 4 | 357.42 | 82.0 | 153.0 | C22H22F3N | Details |
| bio1996 | Tar12 | Toll-like receptor 9 (TLR9) | CHEMBL1346 | DARIFENACIN | Small molecule | Phase 4 | 426.56 | 89.0 | 199.0 | C28H30N2O2 | Details |
| bio1997 | Tar12 | Toll-like receptor 9 (TLR9) | CHEMBL107367 | FARGLITAZAR | Small molecule | Phase 2 | 546.62 | 12.0 | 78.0 | C34H30N2O5 | Details |
| bio1998 | Tar12 | Toll-like receptor 9 (TLR9) | CHEMBL4802233 | ROXATIDINE | Small molecule | Phase 2 | 306.41 | -- | -- | C17H26N2O3 | Details |
| bio1999 | Tar12 | Toll-like receptor 9 (TLR9) | CHEMBL560993 | TIMAPIPRANT | Small molecule | Phase 3 | 348.38 | 41.0 | 998.0 | C21H17FN2O2 | Details |
| bio2000 | Tar12 | Toll-like receptor 9 (TLR9) | CHEMBL2103778 | CILANSETRON | Small molecule | Phase 2 | 319.41 | 35.0 | 44.0 | C20H21N3O | Details |