Bioactive Compounds List
Type Distribution
Max Phase Distribution
Bioactive Compounds List
| Bio ID | Target ID | Target Name | ChEMBL ID | Name | Type | Max Phase | Molecular Weight | Targets | Bioactivities | Molecular Formula | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|
| bio3061 | Tar12 | Toll-like receptor 9 (TLR9) | CHEMBL188462 | ISPRONICLINE | Small molecule | Phase 2 | 234.34 | 17.0 | 42.0 | C14H22N2O | Details |
| bio3062 | Tar12 | Toll-like receptor 9 (TLR9) | CHEMBL1741040 | BQ 788 | Small molecule | Phase 2 | 641.81 | 1.0 | 2.0 | C34H51N5O7 | Details |
| bio3063 | Tar12 | Toll-like receptor 9 (TLR9) | CHEMBL4650220 | ZAVEGEPANT HYDROCHLORIDE | Small molecule | Phase 4 | 675.28 | -- | -- | C36H47ClN8O3 | Details |
| bio3064 | Tar12 | Toll-like receptor 9 (TLR9) | CHEMBL1800159 | RELUGOLIX | Small molecule | Phase 4 | 623.64 | 11.0 | 60.0 | C29H27F2N7O5S | Details |
| bio3065 | Tar12 | Toll-like receptor 9 (TLR9) | CHEMBL5315077 | TILMANOCEPT | Small molecule | Phase 4 | -- | -- | -- | -- | Details |
| bio3066 | Tar12 | Toll-like receptor 9 (TLR9) | CHEMBL2105667 | ORVEPITANT | Small molecule | Phase 2 | 628.63 | 11.0 | 42.0 | C31H35F7N4O2 | Details |
| bio3067 | Tar12 | Toll-like receptor 9 (TLR9) | CHEMBL4297258 | FIRMONERTINIB | Small molecule | Phase 3 | 568.60 | -- | -- | C28H31F3N8O2 | Details |
| bio3068 | Tar12 | Toll-like receptor 9 (TLR9) | CHEMBL197084 | TROFINETIDE | Small molecule | Phase 4 | 315.33 | 7.0 | 23.0 | C13H21N3O6 | Details |
| bio3069 | Tar12 | Toll-like receptor 9 (TLR9) | CHEMBL3889654 | LAROTRECTINIB | Small molecule | Phase 4 | 428.44 | 19.0 | 188.0 | C21H22F2N6O2 | Details |
| bio3070 | Tar12 | Toll-like receptor 9 (TLR9) | CHEMBL4298170 | LERIGLITAZONE HYDROCHLORIDE | Small molecule | Phase 1 | 408.91 | -- | -- | C19H21ClN2O4S | Details |