Bioactive Compounds List
Type Distribution
Max Phase Distribution
Bioactive Compounds List
| Bio ID | Target ID | Target Name | ChEMBL ID | Name | Type | Max Phase | Molecular Weight | Targets | Bioactivities | Molecular Formula | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|
| bio3481 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL5314522 | IRPAGRATINIB | Small molecule | Phase 2 | 570.60 | -- | -- | C28H32F2N6O5 | Details |
| bio3482 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL3544982 | TESEVATINIB TOSYLATE | Small molecule | Unknown | 663.60 | -- | -- | C31H33Cl2FN4O5S | Details |
| bio3483 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL5095247 | EXARAFENIB HYDROCHLORIDE | Small molecule | Phase 1 | 558.05 | -- | -- | C26H35ClF3N5O3 | Details |
| bio3484 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL5095047 | EFROFILCON A | Small molecule | Phase 1 | -- | -- | -- | -- | Details |
| bio3485 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL4802241 | ILUNOCITINIB | Small molecule | Phase 1 | 383.44 | -- | -- | C17H17N7O2S | Details |
| bio3486 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL2108425 | MOBENAKIN | Protein | Phase 2 | -- | -- | -- | -- | Details |
| bio3487 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL5095149 | EFOCIPEGTRUTIDE | Protein | Phase 2 | -- | -- | -- | -- | Details |
| bio3488 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL3039500 | GOLVATINIB TARTRATE | Small molecule | Unknown | 783.79 | -- | -- | C37H43F2N7O10 | Details |
| bio3489 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL2107745 | EFLETIRIZINE DIHYDROCHLORIDE | Small molecule | Unknown | 463.35 | -- | -- | C21H26Cl2F2N2O3 | Details |
| bio3490 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL3039533 | GRAZOPREVIR | Small molecule | Phase 3 | 784.93 | -- | -- | C38H52N6O10S | Details |