Bioactive Compounds List
Type Distribution
Max Phase Distribution
Bioactive Compounds List
| Bio ID | Target ID | Target Name | ChEMBL ID | Name | Type | Max Phase | Molecular Weight | Targets | Bioactivities | Molecular Formula | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|
| bio3571 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL4594381 | DEURUXOLITINIB | Small molecule | Phase 3 | 314.42 | -- | -- | C17H18N6 | Details |
| bio3572 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL1289601 | LENVATINIB | Small molecule | Phase 4 | 426.86 | 335.0 | 389.0 | C21H19ClN4O4 | Details |
| bio3573 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL3643413 | LENIOLISIB | Small molecule | Phase 4 | 450.47 | 126.0 | 300.0 | C21H25F3N6O2 | Details |
| bio3574 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL3039517 | RABUSERTIB | Small molecule | Phase 2 | 436.31 | 312.0 | 329.0 | C18H22BrN5O3 | Details |
| bio3575 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL2103842 | VARLITINIB | Small molecule | Phase 2 | 466.95 | 305.0 | 319.0 | C22H19ClN6O2S | Details |
| bio3576 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL3813842 | PAXALISIB | Small molecule | Phase 2 | 382.43 | 233.0 | 268.0 | C18H22N8O2 | Details |
| bio3577 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL284377 | DEXFOSFOSERINE | Small molecule | Phase 2 | 185.07 | 35.0 | 62.0 | C3H8NO6P | Details |
| bio3578 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL2289112 | TRANS-1,2,3,4,5,6-HEXAHYDROPHTHALOYL-L-THREONINE | Small molecule | -- | 255.27 | 4.0 | 14.0 | C12H17NO5 | Details |
| bio3579 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL2289110 | CIS-1,2,3,4,5,6-HEXAHYDROPHTHALOYL-L-THREONINE | Small molecule | -- | 255.27 | 4.0 | 15.0 | C12H17NO5 | Details |
| bio3580 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL3137334 | LUMINESPIB MESYLATE | Small molecule | Unknown | 579.67 | -- | -- | C27H37N3O9S | Details |