Drug ID:Drug35
Drug Name:Promethazine
CID:4927
DrugBank ID:DB01069
Modality:Small Molecule
Groups:approved
US Approved:YES
Other Approved:YES
Identifier: NCT02765256
Molecular Formula:C17H20N2S
Molecular Weight:284.4 g/mol
Isomeric SMILES:CC(CN1C2=CC=CC=C2SC3=CC=CC=C31)N(C)C
Synonyms:promethazine; Proazamine; Protazine; Promethazin; Prometazin; Vallergine; Dimapp; Fargan; Procit; Promazinamide
Phase 0: 1
Phase 1: 4
Phase 2: 8
Phase 3: 11
Phase 4: 11
Description:A phenothiazine derivative with histamine H1-blocking, antimuscarinic, and sedative properties. It is used as an antiallergic, in pruritus, for motion sickness and sedation, and also in animals. [PubChem]

Molecular Structure

2D Molecular Structure

Knowledge Graph

dtIDCIDCompound NameGene IDGene NameSpeciesPubMed IDsAction
dt325 4927 Promethazine 3269 HRH1 Homo sapiens (human) None
dt326 4927 Promethazine 3356 HTR2A Homo sapiens (human) None
dt327 4927 Promethazine 808 CALM3 Homo sapiens (human) None
dt328 4927 Promethazine 148 ADRA1A Homo sapiens (human) None
dt329 4927 Promethazine 1813 DRD2 Homo sapiens (human) 12476402 None
dt330 4927 Promethazine 3274 HRH2 Homo sapiens (human) 1377455 None
dt331 4927 Promethazine 59340 HRH4 Homo sapiens (human) 11179435 None
dt332 4927 Promethazine 1128 CHRM1 Homo sapiens (human) 12476402 None
dt333 4927 Promethazine 1129 CHRM2 Homo sapiens (human) 12476402 None
dt334 4927 Promethazine 1131 CHRM3 Homo sapiens (human) 12476402 None

  • No data available

Phase Distribution
Phase Description
  • Phase 0: Exploratory trials to assess drug behavior in humans
  • Phase 1: Safety trials to determine safe dosage range
  • Phase 2: Efficacy trials to evaluate therapeutic effects
  • Phase 3: Large-scale trials to confirm efficacy and safety
  • Phase 4: Post-marketing surveillance for long-term safety and efficacy

Trial IDTitlePhaseStatusSponsorIndicationsInterventions
NCT02765256 Fundamental Modification of the Gut Microbiota in the Treatment of Refractory Crohn's Disease PHASE2 COMPLETED University of Pennsylvania Crohn's Disease DRUG: Fluconazole|DRUG: Vancomycin|DRUG: Neomycin… Details

Disease IDDisease NameDefinitionCategoryRelated DrugsMechanism
No data available

Strategy IDTherapeutic StrategySynonymsRelated DrugsMechanism
No data available

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