Target ID:Tar51
ID:P01137
Target Name:Transforming growth factor beta-1 proprotein [Cleaved into: Latency-associated peptide (LAP); Transforming growth factor beta-1 (TGF-beta-1)]
Target Type:Protein
CID:--
URL:https://www.uniprot.org/uniprotkb/P01137
Related Drugs:--

Knowledge Graph

Drug IDDrug NameTypeDrugBank IDTargetsCategoryLatest Progress
No data available

Tissue-Resident T Cells in Chronic Relapsing-Remitting Intestinal Disorders

PMID: 34440651
Year: 2021
Relationship Type: Therapeutic Applications Score: 5.3

Tissue-resident memory T (T(RM)) cells critically contribute to the rapid immunoprotection and efficient immunosurveillance against pathogens, partic…

Post-operative pain after laparoscopic right hemicolectomy for Crohn's disease:…

PMID: 34217174
Year: 2021
Relationship Type: Mechanism Investigation Score: 5.3

AIM: Surgery for Crohn's disease (CD) is characterized by an enhanced inflammatory response. While inflammation can induce hyperalgesia, post-operati…

Vitamin D and Wnt3A have additive and partially overlapping modulatory effects …

PMID: 31147591
Year: 2019
Relationship Type: Mechanism Investigation Score: 5.3

The Wnt/beta-catenin signalling pathway is essential for intestinal epithelium homeostasis, but its aberrant activation is a hallmark of colorectal c…

Ulcer-associated cell lineage expresses genes involved in regeneration and is h…

PMID: 30746716
Year: 2019
Relationship Type: Mechanism Investigation Score: 5.3

Protease inhibition has become a new possible approach in the inflammatory bowel disease (IBD) therapy. A serine exopeptidase, dipeptidyl peptidase …

Glatiramer Acetate Enhances Myeloid-Derived Suppressor Cell Function via Recogn…

PMID: 30068593
Year: 2018
Relationship Type: Mechanism Investigation Score: 5.3

Glatiramer acetate (GA; Copaxone) is a copolymer therapeutic that is approved by the Food and Drug Administration for the relapsing-remitting form of…

Entyvio lengthen dose-interval study: lengthening vedolizumab dose interval and…

PMID: 29727386
Year: 2018
Relationship Type: Therapeutic Applications Score: 5.3

BACKGROUND: Vedolizumab (VDZ), an alpha4beta7 anti-integrin antibody, is efficacious in the induction and maintenance of remission in ulcerative coli…

Overlap syndromes of autoimmune hepatitis: an open question

PMID: 23086110
Year: 2013
Relationship Type: Therapeutic Applications Score: 5.3

The headword "overlap syndromes" of liver diseases includes the coexistence of autoimmune hepatitis, primary biliary cirrhosis, and primary sclerosin…

Crohn's disease genotypes of patients in remission vs relapses after infliximab…

PMID: 23049214
Year: 2012
Relationship Type: Therapeutic Applications Score: 5.3

AIM: To investigate genetic differences between Crohn's disease (CD) patients with a sustained remission vs relapsers after discontinuing infliximab …

Increased suppressor of cytokine signaling-3 expression predicts mucosal relaps…

PMID: 22535619
Year: 2013
Relationship Type: Mechanism Investigation Score: 5.3

BACKGROUND: Most biomarkers predicting mucosal relapse of ulcerative colitis (UC) patients in clinical remission represent low levels of mucosal infl…

Systematic review: management options for primary sclerosing cholangitis and it…

PMID: 21501198
Year: 2011
Relationship Type: Target Validation Score: 5.3

BACKGROUND: Primary sclerosing cholangitis (PSC) remains a challenging disease to manage. The main goals are prevention of disease progression and re…

Overlap, common features, and essential differences in pediatric granulomatous …

PMID: 20683205
Year: 2010
Relationship Type: Mechanism Investigation Score: 5.3

Overlap in the clinical presentation of pediatric granulomatous inflammatory bowel disease may be substantial, depending on the mode of presentation.…

Tilapia head glycolipids reduce inflammation by regulating the gut microbiota i…

PMID: 32219260
Year: 2020
Relationship Type: Mechanism Investigation Score: 5.0

Proton-sensing ovarian cancer G-protein coupled receptor (OGR1) plays an important role in pH homeostasis. Acidosis occurs at sites of intestinal i…

Relapse rates and predictors for relapse in a real-life cohort of IBD patients …

PMID: 30907185
Year: 2019
Relationship Type: Mechanism Investigation Score: 5.0

Gut microbiota has been well recognized in regulation of intestinal homeostasis and pathogenesis of inflammatory bowel diseases. However, the mechan…

Pharmacokinetic Parameters of Infliximab Influence the Rate of Relapse After De…

PMID: 30860594
Year: 2019
Relationship Type: Mechanism Investigation Score: 5.0

Protein tyrosine phosphatases (PTPs) play a critical role in co-ordinating the signaling networks that maintain lymphocyte homeostasis and direct ly…

Candidate IDSource IDSource TypeCompound TypeCandidate NameInclusion Criteria
No data available

Compound IDSource IDSource TypeCompound NameMolecular WeightMolecular FormulaMolecular Species
bio102933 CHEMBL730 Small molecule NITROGLYCERIN 227.08 C3H5N3O9 NEUTRAL Details
bio102934 CHEMBL878 Small molecule METOLAZONE 365.84 C16H16ClN3O3S NEUTRAL Details
bio102935 CHEMBL1079604 Small molecule METAXALONE 221.26 C12H15NO3 NEUTRAL Details
bio102936 CHEMBL1200399 Small molecule BUSPIRONE HYDROCHLORIDE 421.97 C21H32ClN5O2 NEUTRAL Details
bio102937 CHEMBL4297525 Small molecule RELAMORELIN 790.99 C43H50N8O5S BASE Details
bio102938 CHEMBL1200436 Small molecule OXANDROLONE 306.45 C19H30O3 NEUTRAL Details
bio102939 CHEMBL5095183 Small molecule IMLUNESTRANT 524.51 C29H24F4N2O3 NEUTRAL Details
bio102940 CHEMBL1201620 Protein SOMATREM -- -- -- Details
bio102941 CHEMBL1200332 Small molecule PROTRIPTYLINE HYDROCHLORIDE 299.85 C19H22ClN BASE Details
bio102942 CHEMBL3707377 Small molecule SEGESTERONE ACETATE 370.49 C23H30O4 NEUTRAL Details

Strategy IDTherapy StrategySynonymsRelated DrugsMechanism
No data available