Target ID:dt1249
CID:130298939
Compound Name:Eclitasertib
Gene ID:8737
Gene Name:RIPK1
Species:Homo sapiens (human)
PubMed IDs:--
Action:Inhibitor

Knowledge Graph

Target IDCIDCompound NameGene IDGene NameSpeciesAction
dt1198 77108121 (S)-5-benzyl-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-1,2,4-triazole-3-carboxamide 8737 RIPK1 Homo sapiens (human) Inhibition Details
dt1199 77108121 (S)-5-benzyl-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-1,2,4-triazole-3-carboxamide 8737 RIPK1 Homo sapiens (human) Receptor-interacting serine/threonine-protein kinase 1 inhibitor Details
dt1200 77108121 (S)-5-benzyl-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-1,2,4-triazole-3-carboxamide 8737 RIPK1 Homo sapiens (human) Inhibitor Details
dt1201 77108121 (S)-5-benzyl-N-(5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-1H-1,2,4-triazole-3-carboxamide 8737 RIPK1 Homo sapiens (human) Inhibitor Details
dt1247 130298939 Eclitasertib 8737 RIPK1 Homo sapiens (human) Inhibition Details

Drug IDDrug NameTypeDrugBank IDTargetsCategoryLatest Progress
Drug169 SAR443122 Chemical drug -- -- -- Under clinical trials Details

Compound IDSource IDSource TypeCompound NameMolecular WeightMolecular FormulaMolecular Species
No data available

Disease IDDisease NameDefinitionMechanism
No data available

Strategy IDTherapy StrategySynonymsRelated DrugsMechanism
No data available