CMap Candidate Details
Structure:
| CMap ID: | C23735 |
| Pert ID: | BRD-K67075780 |
| Compound Name: | TGX-115 |
| Targets: | -- |
| MoA: | -- |
| SMILES: | Cc1ccccc1Oc2cccc3c(=O)cc([nH]c23)N4CCOCC4 |
| InchiKey: | FWYYZGLCNUZWPF-UHFFFAOYSA-N |
| Compound Aliases: | -- |
| Score ID | Pert ID | Cell Line | Pert Dose | Pert Time | Raw Score (GSE126848) | Normalized Score (GSE126848) | fdr_q_nlog10 (GSE126848) | Raw Score (GSE135251) | Normalized Score (GSE135251) | fdr_q_nlog10 (GSE135251) |
|---|---|---|---|---|---|---|---|---|---|---|
| 8968 | BRD-K67075780 | A375 | 150 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 9222 | BRD-K67075780 | A549 | 150 uM | 6 h | -0.3 | -1.23 | 0.64 | 0.0 | 0.0 | 0.0 |
| 9477 | BRD-K67075780 | AGS | 150 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 9782 | BRD-K67075780 | H1299 | 150 uM | 6 h | 0.24 | 1.01 | 0.12 | 0.0 | 0.0 | 0.0 |
| 10070 | BRD-K67075780 | HA1E | 150 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 10270 | BRD-K67075780 | HCC515 | 150 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 10823 | BRD-K67075780 | HEPG2 | 150 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 10998 | BRD-K67075780 | HT29 | 150 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 11289 | BRD-K67075780 | MCF??7.00 | 150 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 11542 | BRD-K67075780 | NCIH2073 | 150 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 11809 | BRD-K67075780 | NCIH508 | 150 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 12361 | BRD-K67075780 | NOMO1 | 150 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 12455 | BRD-K67075780 | PC3 | 150 uM | 24 h | 0.0 | 0.0 | 0.0 | -0.27 | -0.91 | 0.31 |
| 12842 | BRD-K67075780 | SW480 | 150 uM | 6 h | -0.18 | -0.74 | 0.0 | -0.37 | -1.24 | 1.35 |
| 12963 | BRD-K67075780 | THP1 | 150 uM | 6 h | 0.0 | 0.0 | 0.0 | -0.21 | -0.7 | 0.03 |
| 13327 | BRD-K67075780 | U937 | 150 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 13656 | BRD-K67075780 | VCAP | 150 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |