CMap Candidate Details
Structure:
CMap ID: | C31907 |
Pert ID: | BRD-K93023739 |
Compound Name: | BRD-K93023739 |
Targets: | -- |
MoA: | -- |
SMILES: | Clc1cc(NC(=O)c2cccnc2)c2[nH]c3cnccc3c2c1 |
InchiKey: | JZRMBDHPALEPDM-UHFFFAOYSA-N |
Compound Aliases: | IKK-inhibitor-X |
Score ID | Pert ID | Cell Line | Pert Dose | Pert Time | Raw Score (GSE126848) | Normalized Score (GSE126848) | fdr_q_nlog10 (GSE126848) | Raw Score (GSE135251) | Normalized Score (GSE135251) | fdr_q_nlog10 (GSE135251) |
---|---|---|---|---|---|---|---|---|---|---|
9548 | BRD-K93023739 | AGS | 6.66 uM | 6 h | -0.28 | -1.18 | 0.5 | 0.0 | 0.0 | 0.0 |
9855 | BRD-K93023739 | H1299 | 6.66 uM | 6 h | 0.0 | 0.0 | 0.0 | -0.28 | -0.95 | 0.42 |
9933 | BRD-K93023739 | HA1E | 6.66 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
10313 | BRD-K93023739 | HCC515 | 6.66 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
10881 | BRD-K93023739 | HEPG2 | 6.66 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
11042 | BRD-K93023739 | HT29 | 6.66 uM | 24 h | 0.0 | 0.0 | 0.0 | -0.29 | -0.96 | 0.44 |
11615 | BRD-K93023739 | NCIH2073 | 6.66 uM | 6 h | -0.2 | -0.83 | 0.0 | 0.0 | 0.0 | 0.0 |
11872 | BRD-K93023739 | NCIH508 | 6.66 uM | 6 h | -0.17 | -0.72 | 0.0 | 0.32 | 1.14 | 0.87 |
12172 | BRD-K93023739 | NCIH596 | 6.66 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
12410 | BRD-K93023739 | NOMO1 | 6.66 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
13029 | BRD-K93023739 | THP1 | 6.66 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
13707 | BRD-K93023739 | VCAP | 6.66 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
95863 | BRD-K93023739 | NPC | 10 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
95883 | BRD-K93023739 | MCF??7.00 | 10 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
95942 | BRD-K93023739 | YAPC | 10 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
95955 | BRD-K93023739 | A549 | 10 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
95967 | BRD-K93023739 | PC3 | 10 uM | 6 h | 0.0 | 0.0 | 0.0 | -0.25 | -0.84 | 0.18 |
96849 | BRD-K93023739 | A375 | 3.33 uM | 24 h | -0.23 | -0.95 | 0.09 | 0.0 | 0.0 | 0.0 |