CMap Candidate Details
Structure:
| CMap ID: | C34265 |
| Pert ID: | BRD-U24835547 |
| Compound Name: | GSK-1059615 |
| Targets: | -- |
| MoA: | -- |
| SMILES: | C1=CC2=NC=CC(=C2C=C1C=C3C(=O)NC(=O)S3)C4=CC=NC=C4 |
| InchiKey: | QDITZBLZQQZVEE-UHFFFAOYSA-N |
| Compound Aliases: | -- |
| Score ID | Pert ID | Cell Line | Pert Dose | Pert Time | Raw Score (GSE126848) | Normalized Score (GSE126848) | fdr_q_nlog10 (GSE126848) | Raw Score (GSE135251) | Normalized Score (GSE135251) | fdr_q_nlog10 (GSE135251) |
|---|---|---|---|---|---|---|---|---|---|---|
| 94410 | BRD-U24835547 | A375 | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 94440 | BRD-U24835547 | A549 | 3.33 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 94475 | BRD-U24835547 | ASC | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 94541 | BRD-U24835547 | CD34 | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 94591 | BRD-U24835547 | HCC515 | 0.12 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 94632 | BRD-U24835547 | HEK293 | 0.04 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 94683 | BRD-U24835547 | HELA | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 94735 | BRD-U24835547 | HME1 | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 94785 | BRD-U24835547 | HT29 | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | -0.26 | -0.88 | 0.25 |
| 94828 | BRD-U24835547 | HUVEC | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 94881 | BRD-U24835547 | JURKAT | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 94928 | BRD-U24835547 | MCF10A | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 94968 | BRD-U24835547 | MCF??7.00 | 0.12 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.34 | 1.2 | 1.07 |
| 95008 | BRD-U24835547 | NEU | 3.33 uM | 24 h | -0.27 | -1.11 | 0.37 | 0.0 | 0.0 | 0.0 |
| 95072 | BRD-U24835547 | NPC | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 95112 | BRD-U24835547 | PC3 | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 95154 | BRD-U24835547 | SHSY5Y | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 95232 | BRD-U24835547 | SKL | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | -0.25 | -0.86 | 0.21 |
| 95265 | BRD-U24835547 | THP1 | 10 uM | 24 h | 0.0 | 0.0 | 0.0 | -0.29 | -0.99 | 0.5 |