CMap Candidate Details
Structure:
CMap ID: | C05794 |
Pert ID: | BRD-K10882151 |
Compound Name: | BRD-K10882151 |
Targets: | -- |
MoA: | -- |
SMILES: | O=c1n(Cc2ccccc2)c(/C=C/c3cccnc3)nc4ccccc14 |
InchiKey: | GEKDQXSPTHHANP-OUKQBFOZSA-N |
Compound Aliases: | BO2-inhibits-RAD51 |
Score ID | Pert ID | Cell Line | Pert Dose | Pert Time | Raw Score (GSE126848) | Normalized Score (GSE126848) | fdr_q_nlog10 (GSE126848) | Raw Score (GSE135251) | Normalized Score (GSE135251) | fdr_q_nlog10 (GSE135251) |
---|---|---|---|---|---|---|---|---|---|---|
8911 | BRD-K10882151 | A375 | 40 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
9180 | BRD-K10882151 | A549 | 40 uM | 6 h | -0.22 | -0.9 | 0.05 | -0.24 | -0.81 | 0.13 |
9362 | BRD-K10882151 | AGS | 40 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
9669 | BRD-K10882151 | H1299 | 40 uM | 6 h | -0.25 | -1.03 | 0.2 | 0.2 | 0.73 | 0.03 |
9897 | BRD-K10882151 | HA1E | 40 uM | 24 h | -0.24 | -1.0 | 0.14 | 0.0 | 0.0 | 0.0 |
10275 | BRD-K10882151 | HCC515 | 40 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
10463 | BRD-K10882151 | HCT116 | 40 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
10733 | BRD-K10882151 | HEPG2 | 40 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
10945 | BRD-K10882151 | HT29 | 40 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
11266 | BRD-K10882151 | MCF??7.00 | 40 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
11421 | BRD-K10882151 | NCIH2073 | 40 uM | 6 h | -0.28 | -1.18 | 0.51 | 0.0 | 0.0 | 0.0 |
11712 | BRD-K10882151 | NCIH508 | 40 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.29 | 1.04 | 0.56 |
11989 | BRD-K10882151 | NCIH596 | 40 uM | 6 h | -0.32 | -1.33 | 0.91 | 0.3 | 1.05 | 0.57 |
12269 | BRD-K10882151 | NOMO1 | 40 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
12461 | BRD-K10882151 | PC3 | 40 uM | 24 h | -0.24 | -0.98 | 0.12 | 0.0 | 0.0 | 0.0 |
12733 | BRD-K10882151 | SW480 | 40 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
12971 | BRD-K10882151 | THP1 | 40 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.26 | 0.92 | 0.26 |
13212 | BRD-K10882151 | U937 | 40 uM | 6 h | -0.31 | -1.29 | 0.79 | 0.0 | 0.0 | 0.0 |
13582 | BRD-K10882151 | VCAP | 40 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.22 | 0.79 | 0.07 |