CMap Candidate Details
Structure:
CMap ID: | C07811 |
Pert ID: | BRD-K17140735 |
Compound Name: | SCH-79797 |
Targets: | F2R |
MoA: | Proteasome inhibitor |
SMILES: | CC(C)c1ccc(Cn2ccc3c2ccc4nc(NC5CC5)nc(N)c34)cc1 |
InchiKey: | AVXQPEKZIGPIJW-UHFFFAOYSA-N |
Compound Aliases: | -- |
Score ID | Pert ID | Cell Line | Pert Dose | Pert Time | Raw Score (GSE126848) | Normalized Score (GSE126848) | fdr_q_nlog10 (GSE126848) | Raw Score (GSE135251) | Normalized Score (GSE135251) | fdr_q_nlog10 (GSE135251) |
---|---|---|---|---|---|---|---|---|---|---|
9061 | BRD-K17140735 | A375 | 12 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
9187 | BRD-K17140735 | A549 | 12 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
9375 | BRD-K17140735 | AGS | 12 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
9686 | BRD-K17140735 | H1299 | 12 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
10362 | BRD-K17140735 | HCC515 | 12 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
10475 | BRD-K17140735 | HCT116 | 12 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
10748 | BRD-K17140735 | HEPG2 | 12 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
11116 | BRD-K17140735 | HT29 | 12 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
11272 | BRD-K17140735 | MCF??7.00 | 12 uM | 6 h | -0.21 | -0.85 | 0.01 | 0.0 | 0.0 | 0.0 |
11725 | BRD-K17140735 | NCIH508 | 12 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
12001 | BRD-K17140735 | NCIH596 | 12 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
12595 | BRD-K17140735 | PC3 | 12 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
12747 | BRD-K17140735 | SW480 | 12 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
13228 | BRD-K17140735 | U937 | 12 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
13456 | BRD-K17140735 | VCAP | 12 uM | 24 h | -0.27 | -1.13 | 0.41 | 0.0 | 0.0 | 0.0 |
100157 | BRD-K17140735 | U2OS | 10 uM | 6 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |