CMap Candidate Details
Structure:
| CMap ID: | C09514 |
| Pert ID: | BRD-K22482860 |
| Compound Name: | dalfampridine |
| Targets: | KCNA1; KCNA2; KCNA3; KCNA4; KCNA5; KCNA6; KCNA7; KCNA10; KCNB1; KCNC1; KCNC2; KCNC3; KCND1; KCND2; KCND3; KCNB2 |
| MoA: | Potassium channel blocker |
| SMILES: | Nc1ccncc1 |
| InchiKey: | NUKYPUAOHBNCPY-UHFFFAOYSA-N |
| Compound Aliases: | -- |
| Score ID | Pert ID | Cell Line | Pert Dose | Pert Time | Raw Score (GSE126848) | Normalized Score (GSE126848) | fdr_q_nlog10 (GSE126848) | Raw Score (GSE135251) | Normalized Score (GSE135251) | fdr_q_nlog10 (GSE135251) |
|---|---|---|---|---|---|---|---|---|---|---|
| 121373 | BRD-K22482860 | A375 | 1.11 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 121389 | BRD-K22482860 | HA1E | 3.33 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |
| 121419 | BRD-K22482860 | HELA | 0.125 uM | 24 h | 0.0 | 0.0 | 0.0 | -0.2 | -0.69 | 0.02 |
| 121468 | BRD-K22482860 | MCF??7.00 | 0.125 uM | 24 h | 0.19 | 0.79 | 0.0 | 0.0 | 0.0 | 0.0 |
| 121531 | BRD-K22482860 | YAPC | 0.04 uM | 24 h | 0.24 | 0.99 | 0.09 | 0.0 | 0.0 | 0.0 |
| 129500 | BRD-K22482860 | HT29 | 0.01 uM | 24 h | -0.3 | -1.26 | 0.71 | -0.33 | -1.1 | 0.87 |
| 129564 | BRD-K22482860 | PC3 | 0.08 uM | 24 h | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 | 0.0 |