Bioactive Compounds List
Type Distribution
Max Phase Distribution
Bioactive Compounds List
| Bio ID | Target ID | Target Name | ChEMBL ID | Name | Type | Max Phase | Molecular Weight | Targets | Bioactivities | Molecular Formula | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|
| bio3521 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL4795907 | DARIZMETINIB | Small molecule | Phase 2 | 457.46 | 2.0 | 7.0 | C21H17F2N5O3S | Details |
| bio3522 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL2105742 | VOLASERTIB TRIHYDROCHLORIDE | Small molecule | Unknown | 728.21 | -- | -- | C34H53Cl3N8O3 | Details |
| bio3523 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL1784333 | SERINE AURISTATIN TP | Small molecule | -- | 903.07 | 1.0 | 1.0 | C42H75N6O13P | Details |
| bio3524 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL3962292 | LABUXTINIB | Small molecule | Phase 2 | 377.38 | 1.0 | 2.0 | C20H16FN5O2 | Details |
| bio3525 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL273196 | EFEGATRAN | Protein | Unknown | 416.53 | 23.0 | 100.0 | C21H32N6O3 | Details |
| bio3526 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL16596 | QUIFLAPON | Small molecule | Unknown | 587.19 | 20.0 | 77.0 | C34H35ClN2O3S | Details |
| bio3527 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL261131 | DIACYLGLYCEROL KINASE INHIBITOR II | Small molecule | -- | 489.59 | 269.0 | 566.0 | C28H25F2N3OS | Details |
| bio3528 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL4297329 | PIFUSERTIB | Small molecule | Phase 2 | 424.50 | -- | -- | C26H24N4O2 | Details |
| bio3529 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL603469 | LESTAURTINIB | Small molecule | Phase 3 | 439.47 | 1077.0 | 1794.0 | C26H21N3O4 | Details |
| bio3530 | Tar18 | Serine/threonine-protein kinase cot (COT) | CHEMBL5095383 | RETLIRAFUSP ALFA | Protein | Phase 3 | -- | -- | -- | -- | Details |